Friday, March 27, 2015

Andriol (testosterone undecanoate) - natural male sexual hormone.



Andriol is an oral steroid that produces mild gains and extremely mild unwanted side effects. Unfortunately, it is also an expensive steroid and to make it worthwhile for athletes and bodybuilders to see results from its use, a lot needs to be taken.

Andriol is a unique oral testosterone product, developed by the international drug firm Organon. One of the more recently developed anabolic steroids, Andriol first became available in the early 1980’s. This compound contains 40 mg of Testosterone Undecanoate, based in oil (oleic acid) and sealed inside a capsule. Subtracting the ester weight, this equates to a dosage of approximately 25mg of raw testosterone per cap. The design of this steroid is quite different from that of most oral steroids. Drugs administered orally generally enter the blood stream through the liver. When a steroid compound is given this way without some form of structural protection, it will be quickly broken down during the “first pass”. This process leaves very little steroid intact, basically deactivating the drug. Adding a methyl group (c-17 AA) to the structure is one way to protect it from this process, however stress is also placed on the liver as a result. In some instances this stress can lead to actual damage to liver tissues, so the designers of this steroid sought another way to protect the testosterone molecule. With Andriol, this was accomplished by making a form of testosterone that would be absorbed through the lymphatic system. This is due to its high fat solubility brought about by the ester, and its suspension in oil. Having the compound absorbed this way was thought to be very advantageous, as it allows the steroid to bypass the destructive first-pass through liver. This should permit the compound to enter the blood stream intact, without the need for a harsh chemical alteration.

On paper this drug seems like a great oral testosterone product. Clean, safe and worlds apart from other oral testosterone derivatives like the crude methyltestosterone. But as we always hear in life, if it looks to good to be true, it probably is. There are definitely some issues with Andriol. The first problem is that bioavailability, although clearly worlds apart from trying to take straight testosterone orally, is probably not significant next to c17alpha alkylated orals. Athletes typically find that in doses of less than 240mg per day (6 capsules) effects are generally not seen at all. 240mg of testosterone ester daily, the primary male androgen, and only a meager effect. When doses go higher, maybe 8-10 capsules (320-400mg), new muscle growth is slight to moderate at best, but no incredible bulky gains are ever reported. Logic leads one to believe that only a little testosterone is making its way into circulation. Testosterone is a powerful hormone no matter what the ester or form of administration. If it were active in the blood stream, the results would have to be pronounced. When one injects an oil based testosterone ester like cypionate, a dosage of 400mg per week is more than sufficient to see results. 400mg Andriol per day should be packing on an incredible amount of mass. Where does it all go? Individual problems with absorption may play a role into things here. Clearly there is little to be said except that this drug is unpredictable in its ability to be absorbed and utilized by the body. While one day you might be getting great absorption, perhaps the next day you are getting very little. Studies with men were no better than with women, where again this drug was shown to be unpredictably absorbed and utilized with blood levels ranging from 11.5 to 60.1 nmol/L with 80mg twice daily.

One might also pay interest to the “mildness” of this compound as described by other bodybuilding materials. Andriol is often spoken about as some type of magic product, which to spite being a form of regular testosterone somehow allows for only minimal estrogen conversion. You should know that the way a drug is administered includes a number of factors that can slightly alter its effect, the most predominant being the speed of release. This effects the time it takes for a peak blood level to be reached, and likely the length it takes to see results. The primary reason Testosterone suspension seems more powerful than enanthate is because more drug is active on day one. At the same time estrogen builds up faster and side effects become pronounced very quickly. The ester is also part of the total weight, and 100mg testosterone contains a much larger quantity of testosterone molecules that testosterone plus ester, another reason for varying effect. But these changes do not amount to all that much. The structure of testosterone is what allows it to break down into estrogen. The only way we can really prevent an androgen from converting to estrogen is to change the base molecule, not the ester. Once free in the blood stream we cannot prevent testosterone from being aromatized without interfering with the aromatase enzyme itself. The lack of results and side effects often reported with Andriol must be going hand in hand with poor absorption.

Friday, March 20, 2015

Primobolan - The Ultimate Steroid?


Primobolan Depot is an extremely effective steroid that's earned its respect as the safest injectable steroid. It's the only steroid that will yield solid gains even on a low calorie diet. It's also the only steroid that will build solid muscle slowly with minimal to no side effects... No acne, no aggression, no water bloat, no loss of sex drive, and its the only steroid that will not shut down HPTA (you want to have kids one day right?). I honestly cant think of another steroid that compares to primobolan!

Methenolone is a DHT-based steroid (actually, DHB or dihydroboldenone, the 5-alpha reduced of the milder boldenon). Meaning when it interacts with the aromatase enzyme it does not form estrogens at all.(estrogen is what causes unwanted sides). But unlike Deca Durabolin you do not have to worry about progesterone problems (like bitch tits) either, so now you have the best of both worlds!

Since Primobolan does not convert to estrogen, it displays many favorable characteristics. Estrogen related side effects should not be seen at all when using this steroid. Sensitive individuals need not worry about developing gynecomastia, nor should they notice any water retention with this drug. The gains seen with Primobolan will be only quality muscle mass, and not the smooth bloat which accompanies most steroids open to aromatization. In addition, during a cycle, the user should not have much trouble with blood pressure values, as this effect is also related (generally) to estrogen and water retention - two common side effects that Primobolan just doesn't have.

You will here Primobolan is weaker than deca. That's not exactly accurate. Deca Durabolin is a great substance but is also very calorie dependant. Primobolan is not, Primobolan can allow your diet to be a little loose. A few quotes by Bill Roberts: "It appears to cause less inhibition than Deca Durabolin or testosterone for any given degree of anabolic effect, perhaps because of low CNS activity, lack of conversion to DHT, and lack of aromatization to estrogen." Do you understand what he is saying. Ok this is even true at a range of 600 mgs Primobolan per week which is a highly effective dose. Requiring a little higher dosage to achieve the same anabolic effect, but since it is pleasant to use at doses considerably higher than what is pleasant for nandrolone esters (deca durabolin), it can achieve higher maximum effectiveness. In addition, Primobolan depot is attached to an ester which allows a half-life of about 5 to 10 days. This is a benefit to both the new or veteran user. Every day injections or every other day are a pain in the ass, no pun intended. But every injecting Primo every 5 to 7 days is enough to allow for optimal blood levels.

Primobolan Depot happens to have another plus, the drug is particularly excellent for use as the last injectable in a cycle, since for any given anabolic effect it gives much less inhibition of your natural testosterone production than other steroids such as testosterone, nandrolone, or tren. Therefore, residual levels of Primobolan can allow recovery of your natural test levels as you taper off your cycle while still offering useful anti-catabolic or even anabolic support.

And oh... When people blow up say 30lbs in a cycle its impossible to keep it all as most of it is water bloat. Even if you plan your cycle carefully and do your homework, half your gains, (if not more) will disappear within a few weeks. A slow quality builder like Primobolan allows you to gain for the long term.

Side effects with Primobolan Depot are minimal and manifest themselves only rarely and in persons who are extremely sensitive. Due to the androgenic residual effect, side effects can include light acne, deepening voice or increased hair growth. But who cares? Take B5 for the acne, women love deep voices, and increased hair growth? Cry me a river and shave. Primobolan Depot has even less influence on the liver function than the oral Primobolan so that an increase of the liver's toxin values is extremely unlikely. The blood pressure, cholesterol level, HDL and LDL values, as with Primobolan tablets, usually remain unaffected. Primobolan Depot is generally the safest injectable steroid.

Like the tablets, Primobolan Depot has only a very small influence on the hypothalamuhypophysiat testicular axis so your body's own testosterone production is only reduced when very high dosages are taken over a prolonged period of time.

Stacks: Primobolan is often used in a stack. It is popular for male bodybuilders to stack Primobolan with other steroids in order to obtain a faster and more enhanced effect. Methenolone (Primo) is also one of the rare steroids that works on a reduced calorie diet. This makes Primobolan depot an ideal part of every cutting stack. For dieting (pre contest preparation) Methenolone works best in stack with T3, Clen, Proviron, Deca, and/or Test. During a dieting or cutting phase, a non-aromatizing androgen like Halotestin or trenbolone can be added. The strong androgenic component should help to bring about an added density and hardness to the muscles. On the other hand (or in addition) we could add Winstrol or Anavar, another mild anabolic steroid. The result of this combination should again be a notable increase of muscle mass and hardness, but in this case the gain should not be accompanied by increased side effects. And as mentioned earlier, Primobolan Depot is also used effectively during bulking phases of training. The addition of testosterone, Dianabol or Anadrol prove quite effective for adding new muscle mass. Of course when stacked with those three, we would have to deal with estrogenic side effects, but in such cases Primobolan should allow the user to take a much lower dosage of the more "toxic" drugs and still receive acceptable results.

Friday, March 13, 2015

Effects of Tenbolone on the Body


Trenbolone is a very popular anabolic steroid with stringent side effects, more so than other anabolic steroids. Since it was first developed, Trenbolone has been regarded as a scary, mythic compound. Many people who read about the drug are scared by what they read. The reason is that people don’t understand Trenbolone side effects and the risks compared to the benefits. What you need to understand is that there are numerous other compounds that are much more mysterious than Trenbolone. Once people understand Trenbolone, it’s not as terrifying as they thought.

Review of Trenbolone Side Effects

Trenbolone has some unique side effects to it. Yes, it does have common side effects as any other anabolic steroid but it has its own one-of-a-kind side effects. Bear in mind that some of the unique Trenbolone side effects have made many people to label it a harsh anabolic steroid. Not everyone will experience them but the majority of folks do get them. The side effects people experience will depend on a number of factors:
  • Individual response to compound
  • Lifestyle habits
  • Personal genetics
  • Gender
  • Age
What are some of the adverse side effects you may or may not experience with the use of Trenbolone?

Trenbolone Increases Perspiration

Trenbolone has a tendency to reveal its powerful nutrient partitioning effect. This ability is how every single anabolic steroid works, with some showing it more than others. Trenbolone is one of those anabolic steroids. When this happens, a person can experience a rise in their metabolic rate as an unexpected effect. Excessive sweating can happen any time of the day or night and is often seen at night when a person is sleeping. This side effect isn’t anything real serious or life-threatening but can be a real nuisance. Trenbolone users will need to increase their water intake because the excessive sweating can cause dehydration.

Insomnia and Trouble Falling Asleep

Users of Trenbolone and other anabolic steroids often report suffering with insomnia. While the side effect is minor for many anabolic steroids, Trenbolone users tend to have this side effect much more often. In fact, the number of people who have the side effect is mind-blowing. It’s not known why this happens, but it’s believed its components stimulate the body’s nervous system. This causes people to be unable to sleep, feel tired or continuously get restless sleep (tossing and turning) or constantly wake up during the night. Many Trenbolone acetate or enanthate users need some kind of sleep aid to help them get a good night’s rest. Our recommendations for the best Trenbolone stacks and cycle dosages here.

Gynecomastia Caused by Trenbolone Side Effects

Gynecomastia is a very complicated issue that’s not completely understood. How progesterone and estrogen react with each other is a complex issue. Progestins are seen as inhibitors of Prolactin secretion. There is a significant amount of evidence that claim 19-nor compounds like Nandrolone and Trenbolone can cause the body to generate Prolactn from the pituitary gland.

Trenbolone is a Progestin and acts on the Progestin receptors found in the breast tissue. Both Prolactin and Estrogen receptors are also seen in breast tissue and it’s thought that the Estrogen receptor activity will worsen the progesterone receptor sensitivity. Basically, progestins like Trenbolone will make the estrogen receptor to increase the sensitivity of the estrogen levels and raise the possibility of gynecomastia. Even low levels of estrogen will cause the enlargement of gynecomastia.

The amalgamation of Progesterone, Estrogen and Prolactin will produce an intricate network, which is why gynecomastia is an issue. Prolactin’s effect on this medical condition because of Trenbolone will often show itself in one key way: Nipple lactation – fluid that leaks from the nipples, when pressed or squeezed
Men who have high Prolactin levels could experience Trenbolone side effects like erectile dysfunction and anorgasmia, which is the inability to get an orgasm. There are several ways that people can prevent these problems:
  • Users could use Prolactin-antagonistб which act like dopamine-receptor agonists that reduce or eliminate prolactin levels.
  • Control levels of estrogen by using aromatase inhibitor with compounds that will aromatize like Testosterone or by decreasing testosterone to TRT doses so there is a reduction in aromatization into estrogen.
  • Using vitamin B6 to control the levels of prolactin – 600mg on a daily basis.
It’s important to understand that controlling the levels of estrogen go hand in hand in controlling the levels of prolactin being released by the pituitary glands. However, this won’t work for everyone. Some people still suffer with increases in prolactin even if they have low levels of estrogen while they use Trenbolone. This is why everyone needs to use a Prolactin-antagonist.

Does Tren Decrease Libido?

The problem with one’s libido stems from the increase of Prolactin, and for males this can cause a number of issues:
  • Nipple lactation
  • Reduction in libido
  • Erectile dysfunction
  • Anorgasmia
Keep in mind that progesterone can keep the production of prolactin from occurring and 19-nors like Trenbolone can suppress levels of prolactin. Now, Trenbolone or Nandrolone are considered a progesterone, rather they are anabolic steroids that show signs of progestogenic activity because of the chemical modifications, which is why it’s possible for the hormones to show signs that is contrary to the parent hormone. It’s important people use testosterone while using trenbolone and have another type of prolactin-antagonistic compounds to control the side effects of prolactin.

Trenbolone Cough

Users can experience very mild to extremely serious coughing fits right after getting an injection. Many people feel the rumor is a myth while others view it as a truth. This side effect comes on because of the needle hitting of the capillaries or vein while it’s being injected. When Trenbolone is being injected, it releases an oil-based structure that goes into the ruptured vein and, finally, the bloodstream. What happens is the body is trying to get rid of the foreign substance – it carries the oil to the lungs that the user then coughs out. Thus, the coughing fit ensues! Keep in mind that any oil-based anabolic steroid will cause this side effect. It’s not known why negative side effects of Trenbolone causes a more serious coughing fit than others, although there are several theories as to why this is (some fairly reasonable to others not so much). The coughing fit can be scary to the person experiencing it but hardly ever a life-threatening condition. The intensity of a coughing fit can be very mild – like a tickle in the throat – to serious – full-blown, intense coughing fit. With the more serious coughing fit, people may experience excessive sweating that will stop once the coughing stops.

Cardiovascular Side Effects

Many Trenbolone users say they have experienced a reduction in their pulmonary and cardiovascular capacity while using trenbolone. However, once the users don’t use the drug any longer, the side effect also goes away. It’s believed the side effect is dose-dependent. Many users who use low levels of Trenbolone may not experience this side effect. People who use a higher dose often experience the side effect. What is happening is a bronchial constriction – it makes it hard for the user to suck in copious amounts of oxygen, especially when working out. Of course, everyone is different, so some people will experience it while others will not. This side effect of Trenbolone is not regarded as a serious life-threatening issue, but exercisers may notice issues while they workout. It’s a temporary condition that asthmatic people should understand about, especially if they have a serious asthma attack.

Irritability and Aggression

Trenbolone is just as powerful as androgen as it is an anabolic, with the androgenic strength being five times testosterone’s strength. It’s got 500 androgenic rating, which can increase a user’s feelings of aggression and irritability. Like the above side effect, this is a dose-dependent side effect. The higher the cycle dosage taken, the more likely chance of suffering with the side effect. Some people may not even have this side effect at all. People who have anger problems or a short temper should be careful when using trenbolone because it can increase these traits. It’s advisable that these people do not use Trenbolone to avoid any possible issues. It’s best that only people who have a stable psychological state should use Trenbolone or else the adverse effects on mood may be worse. And, if persons using the drug notice a change in their behavior, they need to be aware of their actions. It all boils down to personal responsibility when people use anabolic steroids or any kind of drug for that matter.

Stress on Kidneys and Liver

One half-truth, half rumor to Trenbolone use is that there is additional stress put on the liver and kidney. Trenbolone isn’t any different than other injectable compounds when it comes to the additional stress but on the human organs. Trenbolone does put a small bit of strain on the liver because of its struggle to hepatic breakdown and metabolism. However, the toxicity of this is hardly an issue. Still, every person needs to take precautions when it comes to their liver and kidney and anybody who has had problems with these organs are advised not to use trenbolone or other anabolic steroids. The kidney damage rumor is from the fact that the urine turns a darker color with a strong rusty orange color to it. It’s often thought to be a bloody urine, which is why people assume it damages the kidneys. Trenbolone side effects don’t cause damage to the kidneys, but it does change the color because it will oxidize.

Trenbolone and the Liver

Trenbolone does not have C-17-alpha alkylation, the chemical modification needed for permit the anabolic steroid oral bioavailability. The modification can show itself in various hepatotoxicity degrees. Trenbolone doesn’t have this feature, but does have a minute amount of hepatotoxicity. This is due to its chemical structure, causing the Trenbolone to have a higher resistance to hepatic breakdown and metabolism.

This minute amount is not a reason to be concerned, for healthy persons, since the liver toxicity doesn’t reach the levels experienced by oral C17-alpha alkylated anabolic steroids. If a person is suffering with pre-existing liver issues, they need to be aware of the problem. Blood work needs to be done on Trenbolone users to keep an eye on the liver enzymes. A doctor may also prescribe a liver support supplement to avoid side effects of Trenbolone from a cycle and to ensure the liver functions properly.

Wednesday, March 4, 2015

Cutting cycle Trenbolone - Primobolan - Winstrol - Masteron.


One of the best ways to get lean is to increase your muscle mass. The more mass on your body, the easier it will be to burn calories and create a deficit which will force your body to pull from its fat stores. An interesting note about body-fat or what scientists like to call, “adipocytes”, is that adipocytes like aromatase. They house it and help produce it. Does that mean the fatter you are, the more estrogen your body will convert from the anabolic steroids you use? Probably.

In any case, body-fat and estrogen are good buddies. We want to disrupt their relationship as much as possible so that we can get both of them to move out of our space. Our rental space where we keep our shredded muscle and veins. After all, muscle just doesn’t look as good when it has layers of fat and water over it. No veins, no sharp division between muscle groups, no abs, no girls and no head turns.

Fat-loss is something I know a tremendous deal about, from both background knowledge from school and applied knowledge on myself, hundreds of clients, and many friends. Fat loss with the aid of juice is something I know even more about.

Alright friends, how do we use juice to help us get shredded. Well, continuing with our point from above about estrogen and body-fat, we want to create an environment and metabolism that has very little of both. Enter non-aromatizing anabolic steroids.

Here are your primary choices:
  • Trenbolone
  • Primobolan
  • Winstrol
  • Masteron
Secondary choices (these drugs sometimes aromatize slightly depending on your genes, but usually not enough to make them inefficient dieting drugs)
  • Halotestin
  • Equipoise
  • Deca Durabolin
The possible drug combinations for a legitimate cutting cycle are numerous. One of the best ways to go about a good cutting cycle is to plan out the weeks ahead. If you are a competitive physique athlete, you know how to do this, if you aren’t this might be a little new.

You can keep some drugs in the program that do aromatize. At least, in the beginning. Lets say you plan on dieting for ten weeks. For the first four, you can still use aromatizing anabolics. You won’t know for sure until you’ve attempted to get lean with drugs a few times over. The less prone you are to estrogenic side affects and water bloat, the longer you can use aromatizing drugs in your cutting arsenal.

If you are very susceptible to these effects, you will have to use non-aromatizing androgens for the entire course along with anti-estrogens in order to maximize the rate and extent of your fat-loss. Nobody wants slow fat loss. Especially when dieting strictly and correctly. We are battling hormones as well as general calories.
In many cases where people have difficulty with estrogen, they have difficulty with fat loss. Whether you are susceptible or not, here is the quickest way to lose body-fat with the assistance of anabolic steroids.

Before we get to the fun stuff, I have to say the diet is precedent over all else. Nutrition is key to getting shredded and it has nothing to do with eating “healthy”.
Okay, fun stuff. First, you need to find your ant-estrogens. I would use at least two, one from each main category, even if you do not typically struggle with water and estrogen while juicing.

My recommendations are Proviron, and Arimidex if you are not susceptible, and if you are, Proviron and Nolvadex.

The difference is that both Proviron and Arimidex will wipe out the aromatase enzyme where Nolvadex occupies the receptor site and blocks the estrogen molecules from hooking up with the receptor. Please see the anti-estrogen page. If you are susceptible, you always have a decent amount of estrogen floating around and you will need a drug that immediately blocks estrogen from wreaking havoc on your physique-Nolvadex.

If you are not susceptible, you just want to make sure that whatever little estrogen you have in your system stays low to non-existent. You do this by taking anti-estrogens that kill the maker of estrogen, the aromatase enzyme. Arimidex is excellent for binding up this enzyme.

Okay, we have our anti-estrogens in place, back to juice. Trenbolone is great. As potent as test and no estrogen or water. Great retention of your hard eared strength and muscle mass as well. Just over 200mg a week of any form should do it. Over 400mg would be unnecessary. Tren usually comes in 75mg strength, give or take a few milligrams. So you will need a minimum of three cc’s a week and upwards of five.

Equipoise is great at around 400mg a week if you are not susceptible to estrogenic effects. With the previous mentioned anti-estrogens, you will probably not have to worry. The Equipose adds a nice vascularity enhancing component to your cycle. Your veins should come out more and more as you get lean and will be accentuated by the Equipose. The nitrogen retaining affect will also help protect your muscle tissue as you add more cardio and decrease your calories.

Anavar works great to aid in strength retention. The more strength you retain while dieting, the less muscle you lose. Anavar has also been shown in studies to specifically aid fat-loss from the intra-abdominal region. It is also associated with an increase in cholesterol profile, raising your HDLs (good cholesterol) and lowering your LDLs (bad cholesterol). Don’t forget the creatine phosphate storage effect of the anavar. This will help keep your muscle bellies a little more full so that you don’t have that flat muscle look as you decrease your carbs. Anavar is a little tough to find sometimes but it is worth it. A decently high dose is needed to get this affect when dieting. At least 15mg and preferably between 20-30mg per day while dieting.

Oral Winstrol is great when dieting if you can afford to take enough. Around 30-50mg per day will greatly enhance your body’s ability to retain muscle at the expense of burning body-fat. Realize, I did not say Winstrol will burn body-fat. It will help shift your metabolism in favor of fat-loss. If you diet well and do your cardio, the Winstrol will aid your body in allowing the deficit of calories to only be pulled from fat, and not muscle.

Realize that there are two orals in this dieting regimen. This is just an example. You can pick any number of combos. Just be sure to give it thought by way of drug mechanism of action, and interaction (synergy) as we’ve said before. The above example is a great cutting regimen for general purposes. Two orals ran together at a sane dosage for ten weeks once or twice a year should be fine on your liver, as long as you are respecting your liver the rest of the year. I am not talking about those who go out drinking three nights a week while trying to get lean. If you are going to do this at all, reserve your liver for filtering drugs that have a purpose.